Compile Data Set for Download or QSAR
Found 104 of ki data for polymerid = 49000362,49000900,49000902
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50018550(1'-Benzyl-3-phenyl-[3,4']bipiperidinyl-2,6-dione |...)copy SMILEScopy InChI
Affinity DataKi:  0.120nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XW4H9QPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM85035(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]PAF from platelet activating factor receptor in human platelets after 3 hrsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P55PWCPubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XW4H9QPubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM82381(L-659,989, (-))copy SMILEScopy InChI
Affinity DataKi:  0.510nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM85035(CAS_65154-06-5 | PAF | bloodplatelet-activatingfac...)copy SMILEScopy InChI
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2610XV6PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50280339((S)-2-[4-(2-Benzenesulfonyl-ethoxy)-3-methoxy-5-(p...)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Compound was evaluated for inhibition of binding of [3H]-C18 PAF to human platelet membrane Platelet activating factor receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50005232((R)-2-{[Acetyl-(2-methoxy-3-octadecylcarbamoyloxy-...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002827(1-{3-(3-Hydroxy-propoxy)-2-propoxy-5-[(2S,5S)-5-(3...)copy SMILEScopy InChI
Affinity DataKi:  1.90nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
LigandPNGBDBM50286012(3-{(R)-7-[1-Dimethylcarbamoyl-6-(4-fluoro-phenyl)-...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Inhibition of platelet activating factor(PAF) by binding to PAF receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46RXM
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002828(1-{3-(3-Morpholin-4-yl-propoxy)-2-propoxy-5-[(2S,5...)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002824((S)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002827(1-{3-(3-Hydroxy-propoxy)-2-propoxy-5-[(2S,5S)-5-(3...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002826(1-{3-(3-Imidazol-1-yl-propoxy)-2-propoxy-5-[(2S,5S...)copy SMILEScopy InChI
Affinity DataKi:  3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  3.20nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)copy SMILEScopy InChI
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NC5ZPRPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002825((R)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002824((S)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:In vitro effect on inhibition of the binding of [3H]C18-Platelet activating factor to human PMN membranes preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002825((R)-5-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-tri...)copy SMILEScopy InChI
Affinity DataKi:  3.72nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50018550(1'-Benzyl-3-phenyl-[3,4']bipiperidinyl-2,6-dione |...)copy SMILEScopy InChI
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XW4H9QPubMed
LigandPNGBDBM50035397(6-(4-Fluoro-phenyl)-3-((R)-3-pyridin-3-yl-1H-pyrro...)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Inhibition of platelet activating factor (PAF) by binding to PAF receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46RXM
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50038766(3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazole-7-carboxy...)copy SMILEScopy InChI
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM39341(11-[(4-methylpiperazin-1-yl)acetyl]-5,11-dihydro-6...)copy SMILEScopy InChI
Affinity DataKi:  5.31nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XW4H9QPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM82381(L-659,989, (-))copy SMILEScopy InChI
Affinity DataKi:  5.48nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:In vitro inhibition of [3H]-C18 PAF binding to human platelet membrane Platelet activating factor receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to PMN membrane receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50038766(3-Pyridin-3-yl-1H-pyrrolo[1,2-c]thiazole-7-carboxy...)copy SMILEScopy InChI
Affinity DataKi:  6.20nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  6.30nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM86231(ATR | ATROPINE | Atropine,(-) | CAS_51-55-8 | CHEM...)copy SMILEScopy InChI
Affinity DataKi:  6.80nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XW4H9QPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM81928(1H,3H-Pyrrolo[1,2-c]thiazole-7-carboxamide,N-(3-be...)copy SMILEScopy InChI
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM81972((S)-(+)-ALPHA-METHYL-1H-IMIDAZOLE-4-ETHANAMINE DIH...)copy SMILEScopy InChI
Affinity DataKi:  9nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM81928(1H,3H-Pyrrolo[1,2-c]thiazole-7-carboxamide,N-(3-be...)copy SMILEScopy InChI
Affinity DataKi:  11.7nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  12.2nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM81972((S)-(+)-ALPHA-METHYL-1H-IMIDAZOLE-4-ETHANAMINE DIH...)copy SMILEScopy InChI
Affinity DataKi:  14.3nMAssay Description:In vitro inhibition of [3H]-C18 PAF binding to human platelet membrane Platelet activating factor receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X588Z
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002829((2S,5S)-2-(3-Methanesulfonyl-5-methoxy-4-propoxy-p...)copy SMILEScopy InChI
Affinity DataKi:  14.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM81930(CAS_129364 | NSC_129364 | RO 19-3704)copy SMILEScopy InChI
Affinity DataKi:  16.9nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)copy SMILEScopy InChI
Affinity DataKi:  17.4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)copy SMILEScopy InChI
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NC5ZPRPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)copy SMILEScopy InChI
Affinity DataKi:  23.2nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM81930(CAS_129364 | NSC_129364 | RO 19-3704)copy SMILEScopy InChI
Affinity DataKi:  38.6nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)copy SMILEScopy InChI
Affinity DataKi:  39.6nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002823(2-{3-Methoxy-2-propoxy-5-[(2S,5S)-5-(3,4,5-trimeth...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Compound was tested for it''s ability to inhibit [3H]C18-PAF binding to human plateletMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7BKP
TargetBeta-arrestin-1(RABBIT)
University of Arizona

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)copy SMILEScopy InChI
Affinity DataKi:  67.4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NC5ZPRPubMed
LigandPNGBDBM50286013((cis)-(2S,3R)-7-[1-Dimethylcarbamoyl-6-(4-fluoro-p...)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Inhibition of platelet activating factor(PAF) by binding to PAF receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46RXM
LigandPNGBDBM50286013((cis)-(2S,3R)-7-[1-Dimethylcarbamoyl-6-(4-fluoro-p...)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Inhibition of platelet activating factor(PAF) by binding to PAF receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S46RXM
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50000714(3-[4-(2-Chloro-phenyl)-9-methyl-6H-1-thia-5,7,8,9a...)copy SMILEScopy InChI
Affinity DataKi:  79.3nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2CJ8BZ8PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50011875(2-Bromo-4-(2-chloro-phenyl)-9-methyl-6H-1-thia-5,7...)copy SMILEScopy InChI
Affinity DataKi:  80.5nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8CC2PubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50366241(CHEMBL297624 | L-652731)copy SMILEScopy InChI
Affinity DataKi:  103nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
TargetPlatelet-activating factor receptor(Homo sapiens (Human))
Broad Institute of MIT and Harvard

Curated by ChEMBL
LigandPNGBDBM50002822((-)-trans 42s,5S)-2-[3-[(2-Oxopropyl)sulfony1]-4-n...)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2445N3BPubMed
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